Local anesthetics and histrionicotoxin are allosteric inhibitors of the acetylcholine receptor. Studies of clonal muscle cells

J Biol Chem. 1982 Jul 25;257(14):8106-8114.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amphibian Venoms / pharmacology*
  • Anesthetics, Local / pharmacology*
  • Animals
  • Carbachol / metabolism
  • Cell Line
  • Clone Cells
  • Dibucaine / pharmacology
  • Kinetics
  • Mathematics
  • Mice
  • Muscles / metabolism*
  • Receptors, Cholinergic / metabolism*
  • Receptors, Nicotinic / drug effects
  • Receptors, Nicotinic / metabolism*

Substances

  • Amphibian Venoms
  • Anesthetics, Local
  • Receptors, Cholinergic
  • Receptors, Nicotinic
  • Carbachol
  • Dibucaine
  • histrionicotoxin